產(chǎn)品屬性:
產(chǎn)品名稱 | Psammaplin A |
規(guī)格 | 100μg |
貨號(hào) | EY-01Y13001 |
Cas No.: 110659-91-1
別名: N/A
化學(xué)名: N/A
分子式: C22H24Br2N4O6S2
分子量: 664.39
溶解度: N/A
儲(chǔ)存條件: N/A
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述:
Psammaplin A, a marine metabolite, is a potent inhibitor of HDAC and DNA methyltransferases. Psammaplin A ia a highly potent and selective DAC1 inhibitor with an IC50 of 0.9 nM. Psammaplin A possess the antimicrobial effect on the Gram-positive bacteria and inhibits DNA synthesis and DNA gyrase activity. Antitumor Activity[1][2].[1]. Matthias G J Baud, et al. Defining the Mechanism of Action and Enzymatic Selectivity of Psammaplin A Against Its Epigenetic Targets. J Med Chem. 2012 Feb 23;55(4):1731-50.
[2]. Psammaplin A, a Natural Bromotyrosine Derivative From a Sponge, Possesses the
特別提醒公司產(chǎn)品僅供科研使用